Zhaomin Xia#, Qiumei Zhu#, Yi Shan, Jiayu Lu, Meidi An, Xiaoxue Mo, Siqi Wang, Wen Yang, Hua Qian, Huaizhen He,Cheng Wang*. MrgX2-targeting ligand screen for antipseudoallergic agents by immobilized His-tag-fused protein technology. Journal of Medicinal Chemistry, 2025, 68(5):5942-5953.
Jiayu Lu#, Zhaomin Xia#, Yongjing Zhang, He Wang, Wen Yang, Siqi Wang, Nan Wang, Yun Liu, Huaizhen He,Cheng Wang*, Langchong He*. "Relative symmetry with electronegativity of different key-groups" strategy for MRGPRX2 antagonist design and its effect on antigen-induced pulmonary inflammation. Acta Pharmaceutica Sinica B, 2025, 15(1): 494-507.
Jiayu Lu, Xin Jia, Yi Shan, Zhaomin Xia, Hua Qian, Siqi Wang, Wen Yang, Wenyu Yang, Delu Che, Xinlei Zhang,Cheng Wang*, Huaizhen He*. Optimization of MrgX2 Antagonists Based on the "Cell Membrane Chromatography-Molecular Docking" Approach. Journal of Medicinal Chemistry, 2025, 68(12): 12531-12543.
Xiaoxue Mo#,Cheng Wang#, Yi Shan, Siqi Wang, Wen Yang, Zhaomin Xia, Zhanguo Qiao, Tao Zhang, Yuanyuan Ding, Rui Liu, Huaizhen He, Langchong He*. Screening and discovery of volatile allergenic components from artemisia ordosica in Yulin region of Northern China. Journal of Hazardous Materials, 2025, 494: 138759.
Jiayu Lu#, Yi Shan#, Na Li, Xiaoxue Mo, Yajing Hou, Delu Che, Fanli Yang, Langchong He,Cheng Wang*, Huaizhen He*. Non-Internalizing Fluorescent Probe targeting mas-related G protein coupled receptor X2: A Tool for Antagonist Screening and Receptor Detection in Blood Samples. ACS Applied Materials & Interfaces, 2025, accept.
Yi Shan, Zhaomin Xia, Meidi An, Wen Yang, Siqi Wang, Fanli Yang, Langchong He,Cheng Wang*, Huaizhen He*. Construction and application of H1R ligand screening materials based on SMA stabilization and his-tag covalent immobilization of membrane proteins. Journal of Chromatography A, 2024, 1729: 465057.
Cheng Wang#, Xiangjun Wang#, Jiayu Lu, Di Wei, Nan Zhou, Youjia Li, Yuanji Wang, Huaizhen He*. Rapid detection of prostate cancer biomarkers in living cells and urine samples using diboronic acid fluorescent probe. Sensors and Actuators B: Chemical, 2023, 392: 134040.
Shuai Ge#,Cheng Wang#, Min Si, Qiumei Zhu, Yi Shan, Na Li, Yawen Wang, Hongliang Wang, Ge Luo, Huaizhen He*, Langchong He*. Site-specific covalent immobilization of SMA-stabilized ACE2 for SARS-CoV-2 recognition and drug screening. ACS Applied Materials & Interfaces, 2023, 15(28): 33348-33361.
Cheng Wang, Tian Hu, Jiayu Lu, Yuexin Lv, Shuai Ge, Yajing Hou, Huaizhen He*. Convenient diaryl ureas as promising anti-pseudo-allergic agents. Journal of Medicinal Chemistry, 2022, 65: 10626-10637.
Yajing Hou#,Cheng Wang#, Jiayu Lu, Min Jia, Yuexin Lv, Xin Jia, Qiumei Zhu, Min Si, Huaizhen He*, Langchong He. Design and synthesis of first environment-sensitive coumarin fluorescent agonists for MrgX2. International Journal of Biological Macromolecules, 2022, 203: 481-491.